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PA24.{1,6} | Bilirubin Metabolism, Jaundice & LFT Interpretation — SDL Guide (Part 2)

Prehepatic Jaundice: Haemolytic Mechanisms

Three-panel diagram showing the bilirubin pathway in prehepatic (haemolytic) jaundice, including the mechanism of UCB accumulation, color-coded laboratory findings, and common causes grouped by haemolytic versus ineffective erythropoiesis.

Prehepatic Jaundice: Mechanism, Lab Pattern, and Causes

Panel A: RBC haemolysis source; unconjugated bilirubin (UCB) in bloodstream; albumin-binding notation; kidney with 'not filtered' marker; liver conjugation step; intestinal urobilinogen cycle; dark stool arrow; urine urobilinogen arrow. Panel B: Rows for total bilirubin, indirect fraction, direct fraction, urine bilirubin (negative), urine urobilinogen (↑↑), stool colour, AST/ALT, ALP, haemoglobin, reticulocytes, LDH, haptoglobin — colour-coded green/orange/red/yellow. Panel C: Haemolytic sub-column: hereditary spherocytosis, G6PD deficiency, sickle cell disease, AIHA (warm/cold), malaria (P. falciparum), transfusion reactions; Ineffective erythropoiesis sub-column: megaloblastic anaemia, thalassaemia.

When RBC destruction accelerates (haemolysis) or erythropoiesis is ineffective, bilirubin production exceeds the conjugation and secretory capacity of normal hepatocytes. The excess remains as unconjugated bilirubin.

Key features of prehepatic jaundice:
- ↑ Total bilirubin, predominantly unconjugated (indirect fraction >80%)
- Urine bilirubin: negative (UCB is albumin-bound; not filtered by the glomerulus)
- Urine urobilinogen: ↑↑ (more CB reaches gut → more urobilinogen formed → more absorbed → more excreted in urine)
- Stool: dark (↑ stercobilin)
- LFT: transaminases normal (no hepatocyte damage), ALP normal
- Blood: ↑ reticulocytes, ↓ haemoglobin, ↑ LDH, ↓ haptoglobin, +/− anaemia

Common causes:
- Hereditary spherocytosis, G6PD deficiency, sickle cell disease
- Autoimmune haemolytic anaemia (warm/cold antibody)
- Malaria (Plasmodium falciparum — hyperparasitaemia → massive haemolysis)
- Transfusion reactions
- Ineffective erythropoiesis: megaloblastic anaemia, thalassaemia (intramedullary destruction)

Hepatic Jaundice: Hepatocellular Injury

Three-panel diagram showing hepatocellular injury: Panel A illustrates a hepatocyte with all three bilirubin-handling steps disrupted (OATP, UGT1A1, MRP2), producing mixed hyperbilirubinaemia; Panel B summarises key lab findings including positive urine bilirubin and elevated AST/ALT; Panel C shows the De Ritis ratio bar chart distinguishing alcoholic from viral hepatitis.

Hepatic (Hepatocellular) Jaundice: Pathophysiology, Lab Pattern, and Clinical Discriminators

Panel A: Portal sinusoid (blood side); OATP transporter (damaged — red X); UCB accumulation back-flux arrow; Hepatocyte nucleus; UGT1A1 conjugation enzyme (reduced — red X); MRP2 canalicular transporter (impaired — red X); Bile canaliculus; Mixed hyperbilirubinaemia label (↑ UCB + ↑ CB); Color legend: UCB (yellow), CB (blue), Biliverdin (green). Panel B: Table rows: Total bilirubin ↑↑ mixed; Urine bilirubin POSITIVE / dark urine icon; Urine urobilinogen variable (early ↑ late ↓); Stool colour pale icon; AST ↑↑↑ / ALT ↑↑↑ / ALP mildly ↑. Panel C: Alcoholic Hepatitis bar (orange, ratio ~2.5); Viral Hepatitis bar (blue, ratio ~0.8); De Ritis Ratio x-axis; Threshold dashed line at 1.0; Annotation: 'AST:ALT > 2:1 → Alcoholic (mitochondrial AST + pyridoxine deficiency)'.

Hepatocellular damage disrupts all three hepatic bilirubin-handling steps simultaneously: uptake (damaged OATP transporters), conjugation (UGT1A1 reduced), and canalicular excretion (MRP2 impaired or canalicular pressure raised by hepatocyte swelling). The result is a mixed hyperbilirubinaemia — both conjugated and unconjugated fractions rise.

Key features of hepatic (hepatocellular) jaundice:
- ↑ Total bilirubin, mixed (both fractions elevated; CB may dominate in severe disease)
- Urine bilirubin: positive (CB is water-soluble and filtered by glomerulus → dark urine)
- Urine urobilinogen: variable (early ↑, late ↓ as liver fails to extract reabsorbed urobilinogen)
- Stool: may be pale (if canalicular excretion severely impaired)
- LFT: markedly ↑ AST and ALT (hepatocyte necrosis → cytosolic enzyme release), ALP mildly to moderately raised
- Synthetic markers: ↓ albumin (chronic), ↑ PT/INR (acute or chronic)

Common causes:
- Viral hepatitis (A, B, C, D, E)
- Alcoholic hepatitis
- Drug-induced liver injury (DILI): paracetamol, anti-TB drugs (isoniazid, rifampicin, pyrazinamide)
- Leptospirosis (Weil disease)
- Autoimmune hepatitis
- Wilson disease (in young patients)

CLINICAL PEARL

The AST:ALT ratio (De Ritis ratio) is a quick discriminator: ratio >2:1 strongly suggests alcoholic hepatitis (mitochondrial AST release + relative pyridoxine deficiency lowering ALT synthesis). Viral hepatitis typically gives AST:ALT ≈1:1 or ALT > AST. However, in advanced cirrhosis of any cause, the ratio may rise as functional hepatocyte mass falls — so interpret in context, not in isolation.

Posthepatic (Obstructive) Jaundice

Three-panel diagram illustrating posthepatic obstructive jaundice: Panel A shows the hepatobiliary pathophysiology with conjugated bilirubin regurgitating into sinusoidal blood due to bile duct obstruction; Panel B summarises clinical consequences including dark urine, pale stools, and pruritus; Panel C classifies extrahepatic and intrahepatic causes.

Posthepatic (Obstructive) Jaundice — Pathophysiology, Clinical Features, and Causes

Panel A: Hepatocyte, Bile canaliculus, Tight junction, Sinusoid, Common bile duct, OBSTRUCTION block (stone/stricture/tumour), Conjugated bilirubin (CB) backflow arrows, 'No CB reaches intestine' marker, Inset LFT bar chart (ALP/GGT markedly elevated; AST/ALT mildly elevated). Panel B: Dark tea-coloured urine flask (Bilirubin +ve, Urobilinogen absent), Pale/clay-coloured acholic stool, Skin cross-section with pruritus/itch marks (bile salt deposition). Panel C: Extrahepatic column — choledocholithiasis (gallstone icon), carcinoma head of pancreas (Courvoisier sign), cholangiocarcinoma, biliary stricture, PSC; Intrahepatic column — PBC (AMA+ve, middle-aged women), Drug-induced cholestasis (chlorpromazine, OCP, anabolic steroids); shared footer: ↑ ALP, ↑ GGT, ↑ conjugated bilirubin in both.

When bile flow is obstructed — whether in the large extrahepatic ducts or in intrahepatic ductules — conjugated bilirubin cannot reach the intestine. It backs up into hepatocyte canaliculi, crosses the tight junctions, and regurgitates into the sinusoidal blood. Because CB is water-soluble, it freely passes into urine.

Key features of posthepatic (obstructive/cholestatic) jaundice:
- ↑ Total bilirubin, predominantly conjugated (direct fraction >50%, often >80%)
- Urine bilirubin: strongly positive → dark 'tea-coloured' urine
- Urine urobilinogen: absent or very low (no CB reaches gut, so no urobilinogen forms)
- Stool: pale/clay-coloured (acholic stools — stercobilin absent)
- Pruritus (bile salt deposition in skin — a key clinical pointer)
- LFT: markedly ↑ ALP and GGT (synthesised by biliary epithelium and released in response to pressure), transaminases mildly to moderately elevated (secondary hepatocyte injury)

Extrahepatic obstruction (large duct):
- Choledocholithiasis (most common in adults — fluctuating jaundice, colicky pain)
- Carcinoma head of pancreas (painless progressive jaundice — Courvoisier sign)
- Cholangiocarcinoma
- Biliary stricture post-surgery or primary sclerosing cholangitis (PSC)

Intrahepatic cholestasis (bile ductule level):
- Primary biliary cholangitis (PBC — AMA positive, middle-aged women)
- Drug-induced cholestasis: chlorpromazine, oral contraceptives, anabolic steroids
- Intrahepatic cholestasis of pregnancy

SELF-CHECK

A 55-year-old woman presents with progressive jaundice for three weeks, pale stools, dark urine, and pruritus. She has no fever, no pain. On examination a non-tender palpable gallbladder is felt (Courvoisier sign). LFT shows total bilirubin 14 mg/dL (direct 12), ALP 620 U/L, GGT 480 U/L, AST 88 U/L, ALT 76 U/L. Which urine finding is most consistent?

A. Urine bilirubin negative, urobilinogen strongly positive

B. Urine bilirubin positive, urobilinogen absent

C. Urine bilirubin negative, urobilinogen absent

D. Urine bilirubin positive, urobilinogen strongly positive

Reveal Answer

Answer: B. Urine bilirubin positive, urobilinogen absent

This is classic posthepatic/obstructive jaundice (carcinoma head of pancreas). Conjugated bilirubin is water-soluble and freely filtered → urine bilirubin is strongly positive (dark urine). Because no CB reaches the intestine, no urobilinogen is formed by colonic bacteria → urobilinogen is absent (not elevated). Option A describes prehepatic jaundice. Option C would require both a non-conjugating liver AND no obstruction — does not match. Option D (both positive) would be seen in severe hepatocellular disease with partial obstruction.